Indian Patents
Title of Invention

PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR ALPHA AGONIST COMPOUNDS.
Abstract The present invention is directed to compounds represented by the following structural formula, and pharmaceutically acceptable salts, solvates and hydrates thereof, R1 is a substituted or unsubstituted group selected from C1-C8 alkyl, aryl-CO-2-alkyl, heteroaryl-CO-2-alkyl, C3-C6 cycloalkylaryl-CO-2-alkyl or phenyl. W is O or S. R2 is H or a substituted or unsubstituted group selected from C1-C6 alkyl, C3-C6 cycloalkyl and heteroaryl. X is a C2-C5 alkylene linker wherein one carbon atom of the linker may be replaced with O, NH or S. Y is C, O, S, NH or a single bond. Furthermore, E is (CH2)nCOOH, wherein n is 0, 1, 2 or 3, or C(R3)(R4)A, wherein A is an acidic functional group such as carboxyl, carboxamide substituted or unsubstituted sulfonamide, or substituted or unsubstituted tetrazole. R3 is H, saturated or unsaturated C1-C5 alkyl, C1-C5 alkoxy. Additionally, R4 is H, halo, a substituted or unsubstituted group selected from C1-C5 alkyl, C1-C5 alkoxy, C3-C6 cycloalkyl, arylCO-C4alkyl and phenyl, or R3 and R4 are combined to form a C3-C4 cycloalkyl.
Full Text

Documents:

278-kolnp-2003-granted-abstract.pdf

278-kolnp-2003-granted-claims.pdf

278-kolnp-2003-granted-correspondence.pdf

278-kolnp-2003-granted-description (complete).pdf

278-kolnp-2003-granted-form 1.pdf

278-kolnp-2003-granted-form 13.pdf

278-kolnp-2003-granted-form 2.pdf

278-kolnp-2003-granted-form 26.pdf

278-kolnp-2003-granted-form 3.pdf

278-kolnp-2003-granted-form 5.pdf

278-kolnp-2003-granted-gpa.pdf

278-kolnp-2003-granted-letter patent.pdf

278-kolnp-2003-granted-reply to examination report.pdf

278-kolnp-2003-granted-specification.pdf

278-kolnp-2003-granted-translated copy of priority document.pdf


« Previous Patent
Next Patent »
Patent Number 217445
Indian Patent Application Number 278/KOLNP/2003
PG Journal Number 13/2008
Publication Date 28-Mar-2008
Grant Date 26-Mar-2008
Date of Filing 06-Mar-2003
Name of Patentee ELI LILLY AND COMPANY
Applicant Address LILLY CORPORATE CENTER, DC 1104, INDIANAPOLIS, IN 46285
Inventors:
# Inventor's Name Inventor's Address
1 1] MANTLO, NATHAN, BRYAN 7325 EAST 800 NORTH, BROWNSBURG, IN 46112
2 2] COLLADO CANO, IVAN LILLY S.A., AVDA. INDUSTRIA, 30, E-28108 ALCOBENDAS-MADRID
3 3] DOMINIANNI, SAMUEL, JAMES 7873 CLEARWATER COVE DRIVE, INDIANAPOLIS, IN 46240
4 4] ETGEN, GARRET, JAY, JUNIOR 13763 ADIOS PASS, CARMEL, IN 46032
5 5] GARCIA-PAREDES, CRISTINA LILLY S.A., AVDA. INDUSTRIA, 30, E-28108 ALCOBENDAS-MADRID
6 6] JOHNSTON, RICHARD, DUANE 2712 FOREST LANE, GREENFIELD, IN 46140
7 7] LETOURNEAU, MICHAEL, EDWARD 6024 MCCLELLAN COURT, INDIANAPOLIS, LIN 46254
8 8] MARTINELLI, MICHAEL, JOHN 1935 MULSANNE DRIVE, ZIONSVILLE, IN 46077
9 9] MAYHUGH, DANIEL, RAY 9681 TROON COURT, CARMEL, IN 46032
10 10] SAEED, ASHRAF 1500 WORCESTER ROAD, APARTMENT 428, FRAMINGHAM, MA 01702
11 11] THOMPSON, RICHARD, CRAIG 763 NORTH 900 WEST, FRANKFORT, IN 46041
12 12] WANG, XIADONG 14066 HONEY TREE DRIVE, CARMEL, IN 46032
13 13] COFFEY, DAVID, SCOTT 6246 TENNISON WAY, INDIANAPOLIS, IN 46236
14 14] SCHMID, CHRISTOPHER, RANDALL 6235 CENTRAL AVENUE, INDIANAPOLIS, IN 46220
15 15] VICENZI, JEFFREY, THOMAS 49 TIMBER LANE, BROWNSBURG, IN 46112
16 16] XU, YANPING 13832 BARNETT PLACE, FISHERS, IN 46038
PCT International Classification Number C 07 D 249/12
PCT International Application Number PCT/US01/42928
PCT International Filing date 2001-11-09
PCT Conventions:
# PCT Application Number Date of Convention Priority Country
1 60/247,317 2000-11-10 U.S.A.