| Title of Invention | " PEPTIDYL ANALOGS ACTIVE AT THE GTROWTH HORMONE SECDRETGOGUE RECEPTOR" |
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| Abstract | Disclosed are peptide and peptidomimetic compounds generally according to formula (I), and pharmaceutically acceptable salts thereof, that are useful as GHRP analogs: R1-A2-A3-A4-A5-R2 (I) or a pharmaceutically acceptable salt thereof, wherein: A1 is Aib, Apc or Inp; A2 is D-Bal, D-Bip, D-Bpa, D-Dip, D-1Nal, D-2Na1, D-Ser(Bzl), or D-Trp; A3 is D-Bal, D-Bip, D-Bpa, D-Dip, D-1Nal, D-2Nal, D-Ser(Bzl), or D-Trp; A4 is 2Fua, Orn, 2Pa1, 3Pal, 4Pa1, Pff, Phe, Pim, Taz, 2Thi, 3Thi, Thr(Bzl); A5 is Apc, Dab, Dap, Lys, Orn, or deleted; R1 is hydrogen, (C1-6)alkyl, (C5-14)aryl, (C1-6)alkyl(C5-14)aryl, (C3-8)cycloakyl, or (C2-10)acyl; and R2 is OH or NH2; and pharmaceutical compositions and methods of use thereof. (FIG. - Nil) |
| Full Text |
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1973-kolnp-2004-granted-abstract.pdf
1973-kolnp-2004-granted-assignment.pdf
1973-kolnp-2004-granted-claims.pdf
1973-kolnp-2004-granted-correspondence.pdf
1973-kolnp-2004-granted-description (complete).pdf
1973-kolnp-2004-granted-examination report.pdf
1973-kolnp-2004-granted-form 1.pdf
1973-kolnp-2004-granted-form 13.pdf
1973-kolnp-2004-granted-form 18.pdf
1973-kolnp-2004-granted-form 3.pdf
1973-kolnp-2004-granted-form 5.pdf
1973-kolnp-2004-granted-gpa.pdf
1973-kolnp-2004-granted-letter patent.pdf
1973-kolnp-2004-granted-reply to examination report.pdf
1973-kolnp-2004-granted-specification.pdf
| Patent Number | 220273 | ||||||||
|---|---|---|---|---|---|---|---|---|---|
| Indian Patent Application Number | 01973/KOLNP/2004 | ||||||||
| PG Journal Number | 21/2008 | ||||||||
| Publication Date | 23-May-2008 | ||||||||
| Grant Date | 21-May-2008 | ||||||||
| Date of Filing | 21-Dec-2004 | ||||||||
| Name of Patentee | SOCIETE DE CONSEIL DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES S.A.S. | ||||||||
| Applicant Address | 51-53, RUE DU DOCTEUR BALANCHE, FRANCE. | ||||||||
Inventors:
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| PCT International Classification Number | A61K38/40 | ||||||||
| PCT International Application Number | PCT/US2003/024834 | ||||||||
| PCT International Filing date | 2003-08-08 | ||||||||
PCT Conventions:
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