Title of Invention

ANTI-INFLAMMATORY 17, BETA-CARBOTHIOATE ESTER DERIVATIVES OF ANDROSTANE WITH A CYCLIC ESTER GROUP IN POSITION 17. ALPHA

Abstract There are provided compound of formula (I) wherein R1 represents C1-6 alkyl or C1-6 haloalkyl; R2 represents C3-8 cycloalkyl or C3-8 cycloalkenyl either of which may optionally be substituted by one or more groups selected from oxo, methyl, methylene and halogen; R3 UHSUHVHQWVK\GURJHQPHWK\O ZKLFKPD\EHLQHLWKHUWKH.RUconfiguration) or methylene; R4 and R5 are the same or different and each represents hydrogen or halogen; and (AA) represents a single or a double bond; and solvates thereof, processes for preparing them and their use in therapy (FIG. - nil
Full Text

Documents:

1495-kolnp-2003-granted-abstract.pdf

1495-kolnp-2003-granted-assignment.pdf

1495-kolnp-2003-granted-claims.pdf

1495-kolnp-2003-granted-description (complete).pdf

1495-kolnp-2003-granted-examination report.pdf

1495-kolnp-2003-granted-form 1.pdf

1495-kolnp-2003-granted-form 13.pdf

1495-kolnp-2003-granted-form 18.pdf

1495-kolnp-2003-granted-form 3.pdf

1495-kolnp-2003-granted-form 5.pdf

1495-kolnp-2003-granted-gpa.pdf

1495-kolnp-2003-granted-letter patent.pdf

1495-kolnp-2003-granted-reply to examination report.pdf

1495-kolnp-2003-granted-specification.pdf


Patent Number 221126
Indian Patent Application Number 01495/KOLNP/2003
PG Journal Number 25/2008
Publication Date 20-Jun-2008
Grant Date 18-Jun-2008
Date of Filing 18-Nov-2003
Name of Patentee GLAXO GROUP LIMITED
Applicant Address GLAXO WELLCOME HOUSE,BERKELEY AVENUE,GREENFORD, MIDDLESEX, UB6 0NN
Inventors:
# Inventor's Name Inventor's Address
1 BIGGADIKE KEITH GLAXOSMITHKLINE, GUNNELS WOOD ROAD, STEVENAGE HERTFORDSHIRE, SG1 2NY
2 JONES PAUL GLAXOSMITHKLINE, GUNNELS WOOD ROAD, STEVENAGE HERTFORDSHIRE, SG1 2NY
3 PAYNE JEREMY JOHN GLAXOSMITHKLINE, GUNNELS WOOD ROAD, STEVENAGE HERTFORDSHIRE, SG1 2NY
PCT International Classification Number C07J 31/00
PCT International Application Number PCT/GB02/01971
PCT International Filing date 2002-04-30
PCT Conventions:
# PCT Application Number Date of Convention Priority Country
1 0127988.4 2001-11-22 U.K.
2 0110578.2 2001-04-30 U.K.
3 0202637.5 2002-02-05 U.K.
4 0202442.0 2002-02-02 U.K.