Title of Invention

1,2,3-TRISUBSTITUTED ARYL AND HETEROARYL DERIVATIVES AS MODULATORS OF METABOLISM AND THE PROPHYLAXIS AND TREATMENT OF DISORDERS RELATED THERETO SUCH AS DIABETES AND HYPERGLYCEMIA

Abstract The present invention relates to certain 1,2,3-trisubstituted aryl and heteroaryl derivatives of Formula (Ia) that are modulators of metabolism. Accordingly, compounds of the present invention are useful in the prophylaxis or treatment of metabolic disorders and complications thereof, such as, diabetes and obesity.
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01150-kolnp-2005-abstract.pdf

01150-kolnp-2005-claims.pdf

01150-kolnp-2005-description complete.pdf

01150-kolnp-2005-drawings.pdf

01150-kolnp-2005-form 1.pdf

01150-kolnp-2005-form 3.pdf

01150-kolnp-2005-form 5.pdf

01150-kolnp-2005-international publication.pdf

1150-kolnp-2005-granted-abstract.pdf

1150-kolnp-2005-granted-assignment.pdf

1150-kolnp-2005-granted-claims.pdf

1150-kolnp-2005-granted-correspondence.pdf

1150-kolnp-2005-granted-description (complete).pdf

1150-kolnp-2005-granted-drawings.pdf

1150-kolnp-2005-granted-examination report.pdf

1150-kolnp-2005-granted-form 1.pdf

1150-kolnp-2005-granted-form 13.pdf

1150-kolnp-2005-granted-form 18.pdf

1150-kolnp-2005-granted-form 3.pdf

1150-kolnp-2005-granted-form 5.pdf

1150-kolnp-2005-granted-gpa.pdf

1150-kolnp-2005-granted-letter patent.pdf

1150-kolnp-2005-granted-reply to examination report.pdf

1150-kolnp-2005-granted-sequence listing.pdf

1150-kolnp-2005-granted-specification.pdf

abstract-01150-kolnp-2005.jpg


Patent Number 222137
Indian Patent Application Number 01150/KOLNP/2005
PG Journal Number 30/2008
Publication Date 25-Jul-2008
Grant Date 23-Jul-2008
Date of Filing 15-Jun-2005
Name of Patentee ARENA PHARMACEUTICALS INC.
Applicant Address 6166 NANCY RIDGE DRIVE, SAN DIEGO, CA 92121-3223
Inventors:
# Inventor's Name Inventor's Address
1 JONES ROBERT M 10937 CORTE LUZ DEL SOL, SAN DIEGO, CALIFORNIA 92130
2 SEMPLE GRAEME 15920 CAMINO CODORNIZ, SAN DIEGO, CALIFORNIA 92127
3 FIORAVANTI BEATRIZ 60 WEST STONE LOOP, NO. 327 TUCSON, ARIZONA 85704
4 PEREIRA GUILHERME 7366 MESA COLLEGE DRIVE, NO. 43 SAN DIEGO, CALIFORNIA 92111
5 CALDERON IMELDA 10971 CAMINITO ARCADA, SAN DIEGO, CALIFORNIA 92131
6 UY JANE 510A SOUTH MADISON AVENUE, MONROVIA, CALIFORNIA 91016
7 DUVUURI KAMESHWARI 2301 THE WOODS LANE, LEXINGTON, KENTUCKY 40502
8 CHOI JIN SUN KAROLINE 9926 SCRIPPS WESTVIEW WAY, NO. 251, SAN DIEGO, CALIFORNIA 92131
9 XIONG YIFENG 5036 PEARLMAN WAY, SAN DIEGO, CALIFORNIA 92130
10 DAVE VIBHA 6188 SUNSET CREST WAY, SAN DIEGO, CALIFORNIA 92121
PCT International Classification Number C07D 401/14
PCT International Application Number PCT/US2004/001267
PCT International Filing date 2004-01-14
PCT Conventions:
# PCT Application Number Date of Convention Priority Country
1 60/440,394 2003-01-14 U.S.A.
2 60/453,390 2003-03-06 U.S.A.
3 60/449,829 2003-02-24 U.S.A.
4 60/470,875 2003-05-14 U.S.A.