Title of Invention

CHIRAL 1,4-DISUBSTITUTED PIPERAZINES PROCESS FOR THEIR PREPARATION AND INTERMEDIATES

Abstract The invention discloses a process for the stereoselective preparation of a compound of formula III wherein R and R' each independently represents a C1-C3 alkyl group; Ar represents dihydro-benzodioxinyl or benzodioxinyl, or phenyl optionally substituted with up to three substituents independently selected from halogen, methoxy, halomethyl, dihalomethy and trihalomethyl. The invention also discloses a compound of formula IV wherein Ar and R are as defined above obtained by reduction of the compound of formula III, process for their preparation and intermediates.
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Documents:

1338-kolnp-2004-granted-abstract.pdf

1338-kolnp-2004-granted-assignment.pdf

1338-kolnp-2004-granted-claims.pdf

1338-kolnp-2004-granted-correspondence.pdf

1338-kolnp-2004-granted-description (complete).pdf

1338-kolnp-2004-granted-examination report.pdf

1338-kolnp-2004-granted-form 1.pdf

1338-kolnp-2004-granted-form 18.pdf

1338-kolnp-2004-granted-form 3.pdf

1338-kolnp-2004-granted-form 5.pdf

1338-kolnp-2004-granted-gpa.pdf

1338-kolnp-2004-granted-letter patent.pdf

1338-kolnp-2004-granted-reply to examination report.pdf

1338-kolnp-2004-granted-specification.pdf


Patent Number 222139
Indian Patent Application Number 01338/KOLNP/2004
PG Journal Number 30/2008
Publication Date 25-Jul-2008
Grant Date 23-Jul-2008
Date of Filing 10-Sep-2004
Name of Patentee WYETH
Applicant Address FIVE GIRALDA FARMS, MADISON, NJ 07940-0874
Inventors:
# Inventor's Name Inventor's Address
1 JIRKOVSKY IVO P.O. BOX 1209, WAITSFIELD, VT 05673
2 ZELDIS JOSEPH 195 LONG CLOVE ROAD, NEW CITY, NY 10956
3 FEIGELSON GREGG BRIAN ONE INDEPENDENCE LANE, MONSEY, NY 10952
PCT International Classification Number C07D 401/00
PCT International Application Number PCT/US03/07176
PCT International Filing date 2003-03-10
PCT Conventions:
# PCT Application Number Date of Convention Priority Country
1 60/363,458 2002-03-12 U.S.A.