Title of Invention | CHEMICAL COMPOUNDS CONTAINING TOCOPHEROL AND AT LEAST ONE ADDITIONAL PHARMACEUTICAL ACTIVE SUBSTANCE |
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Abstract | The invention relates to chemical compounds in the form of their racemates, enantiomers or diastereomers with general formula I in which R stands for the unchanged portion of a variable pharmaceutical active ingredient molecule, B stands for a spacer, and Toc with the formula and R', R" and R''' are equal to H or methyl stands for tocopherol and A stands for C=X, SOm, X or CH2, whereby X is equal to 0, S or NR1 (when n 1) or S or NR1 (when n = 0), and B means a grouping X-R2-Y with Y equal to C=X, SOm or C(XR3)R4, and n is equal to 0 to 6, preferably 0, 1, 2 or 3, and m stands for 1 or 2, whereby R1 stands for H, C1 to C10-alkyl, preferably C1 to C6-alkyl or aryl, Het or an aryl or Het radical that is bonded via a C1 to C6-spacer, preferably C1 to C3, and whereby R2 is selected from the group alkylene, arylene or Het spacers as well as combinations thereof, whereby the latter are linked to one another either directly or via radical A or via grouping X0-A-Xp, whereby o and p are equal to 0, 1 or 2, and the latter can be the same or different, and whereby R3 and R4 stand for H, C1 to C10-alkyl, preferably C1-C6-alkyl or aryl, Het or an aryl or Het radical that is bonded via a C1 to C6 spacer, preferably C1 to C3-spacers. |
Full Text |
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00392-kolnp-2005 correspondence.pdf
00392-kolnp-2005 correspondence_1.1.pdf
00392-kolnp-2005 correspondence_1.2.pdf
00392-kolnp-2005 correspondence_1.3.pdf
00392-kolnp-2005 description(complete).pdf
00392-kolnp-2005 international publication.pdf
00392-kolnp-2005 international search authority report.pdf
00392-kolnp-2005 pct others.pdf
00392-kolnp-2005 priority document.pdf
392-kolnp-2005-granted-abstract.pdf
392-kolnp-2005-granted-assignment.pdf
392-kolnp-2005-granted-claims.pdf
392-kolnp-2005-granted-correspondence.pdf
392-kolnp-2005-granted-description (complete).pdf
392-kolnp-2005-granted-examination report.pdf
392-kolnp-2005-granted-form 1.pdf
392-kolnp-2005-granted-form 13.pdf
392-kolnp-2005-granted-form 18.pdf
392-kolnp-2005-granted-form 3.pdf
392-kolnp-2005-granted-form 5.pdf
392-kolnp-2005-granted-gpa.pdf
392-kolnp-2005-granted-letter patent.pdf
392-kolnp-2005-granted-reply to examination report.pdf
392-kolnp-2005-granted-specification.pdf
Patent Number | 222157 | |||||||||
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Indian Patent Application Number | 392/KOLNP/2005 | |||||||||
PG Journal Number | 30/2008 | |||||||||
Publication Date | 25-Jul-2008 | |||||||||
Grant Date | 23-Jul-2008 | |||||||||
Date of Filing | 10-Mar-2005 | |||||||||
Name of Patentee | JSW-RESEARCH FORSCHUNGSLABOR GMBH | |||||||||
Applicant Address | RANKENGASSE 28, A-8020 GRAZ | |||||||||
Inventors:
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PCT International Classification Number | C07D 405/12 | |||||||||
PCT International Application Number | PCT/AT2004/000234 | |||||||||
PCT International Filing date | 2004-07-01 | |||||||||
PCT Conventions:
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