Title of Invention | A PROCESS FOR PREPARING OPTICALLY PURE (S,S)-2-(3-CHLOROPHENYL)-3,5,5-TRIMETHYL-2-MORPHOLINOL |
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Abstract | The present invention relates to a process for preparing optically enriched (S,S)-hydroxybupropion, or a phannaceutically acceptable salt thereof, comprising: (a) contacting hydroxybupropion with optically pure camphoric acid, tartaric acid, malic acid or mandelic acid; or an optically pure derivative thereof: (b) isolating an optically enriched salt of (S,S)-hydroxybupropion; and (c) contacting the salt of (S,S)-hydroxybupropion with a base. |
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in-pct-2002-1487-che abstract.pdf
in-pct-2002-1487-che claims granted.pdf
in-pct-2002-1487-che correspondence others.pdf
in-pct-2002-1487-che correspondence po.pdf
in-pct-2002-1487-che descripetion (complete) granted.pdf
in-pct-2002-1487-che petition.pdf
in-pct-2002-1487-che power of attorney.pdf
Patent Number | 226987 | ||||||||||||
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Indian Patent Application Number | IN/PCT/2002/1487/CHE | ||||||||||||
PG Journal Number | 07/2009 | ||||||||||||
Publication Date | 13-Feb-2009 | ||||||||||||
Grant Date | 31-Dec-2008 | ||||||||||||
Date of Filing | 19-Sep-2002 | ||||||||||||
Name of Patentee | SEPRACOR INC | ||||||||||||
Applicant Address | 111 LOCKE DRIVE, MARLBOROUGH, MA 01752, | ||||||||||||
Inventors:
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PCT International Classification Number | A61K31/5375 | ||||||||||||
PCT International Application Number | PCT/US00/23080 | ||||||||||||
PCT International Filing date | 2000-08-23 | ||||||||||||
PCT Conventions:
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