Title of Invention | NOVEL DIPEPTIDYL PEPTIDASE IV INHIBITORS, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
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Abstract | The present invention relates to novel antidiabetic, hypolipidemic, and anticholesteromic, antiobesity compounds representated by formula I, where R,Rl,R2,R3,A,B,m,n are as defined ,their derivatives, their analogs, their tautomeric forms, their stereoisomers, their diastereomers , their bioisosteres, their polymorphs, their pharmaceutically acceptable salts and pharmaceutically acceptable compositions containing them. More specifically, the present invention relates to compounds of the general formula I which are predominantly serine protease inhibitors, particularly dipeptidyl peptidase inhibitors, more particularly dipeptidyl peptidase IV inhibitors, their derivatives, their analogs, their tautomeric forms, their stereoisomers, their diastereomers , their bioisosteres, their polymorphs, their pharmaceutically acceptable salts and pharmaceutically acceptable compositions containing them. The present invention also relates to the processes for the preparation of novel compounds of formula I and novel intermediates and also their use as antidiabetic, hypolipidemic, anticholesteromic and antiobesity compounds |
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610 -che-2006-correspondance-others.pdf
610 -che-2006-correspondance-po.pdf
610 -che-2006-description provisional.pdf
610-CHE-2006 AMENDED CLAIMS 19-12-2011.pdf
610-CHE-2006 AMENDED CLAIMS 29-09-2011.pdf
610-CHE-2006 CORRESPONDENCE OTHERS 15-09-2011.pdf
610-CHE-2006 CORRESPONDENCE OTHERS 19-12-2011.pdf
610-CHE-2006 EXAMINATION REPORT REPLY RECEIVED 29-09-2011.pdf
610-CHE-2006 FORM-1 29-09-2011.pdf
610-CHE-2006 FORM-13 29-09-2011.pdf
610-CHE-2006 FORM-3 15-09-2011.pdf
610-CHE-2006 FORM-3 29-09-2011.pdf
610-CHE-2006 OTHER PATENT DOCUMENT 15-09-2011.pdf
610-CHE-2006 CORRESPONDENCE OTHERS 10-02-2012.pdf
610-CHE-2006 CORRESPONDENCE OTHERS 15-09-2011.pdf
610-CHE-2006 CORRESPONDENCE OTHERS 20-02-2012.pdf
610-CHE-2006 CORRESPONDENCE OTHERS.pdf
610-CHE-2006 CORRESPONDENCE PO.pdf
610-CHE-2006 CORRESPONDENCE. OTHERS 20-02-2012.pdf
610-che-2006 description (complete) 27-03-2007.pdf
610-CHE-2006 FORM-13 10-02-2012.pdf
610-CHE-2006 FORM-3 15-09-2011.pdf
610-CHE-2006 FORM-3 16-07-2012.pdf
610-CHE-2006 POWER OF ATTORNEY.pdf
610-CHE-2006 CORRESPONDENCE-OTHERS 21-10-2009.pdf
610-che-2006 correspondene others 14-08-2007.pdf
Patent Number | 251197 | |||||||||||||||
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Indian Patent Application Number | 610/CHE/2006 | |||||||||||||||
PG Journal Number | 09/2012 | |||||||||||||||
Publication Date | 02-Mar-2012 | |||||||||||||||
Grant Date | 29-Feb-2012 | |||||||||||||||
Date of Filing | 03-Apr-2006 | |||||||||||||||
Name of Patentee | MATRIX LABORATORIES LTD. | |||||||||||||||
Applicant Address | 1-1-151/1, IV FLOOR, SAIRAM TOWERS, ALEXANDER ROAD SECUNDERABAD 500 003 | |||||||||||||||
Inventors:
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PCT International Classification Number | C07D401/12 | |||||||||||||||
PCT International Application Number | N/A | |||||||||||||||
PCT International Filing date | ||||||||||||||||
PCT Conventions:
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