Title of Invention | NOVEL TRIAZOLE DERIVATIVES RECEPTORS |
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Abstract | The present invention provides novel triazole derivatives as ghrelin analogue ligands of growth hormone secretagogue receptors according to formula (I) that are useful in the treatment or prophylaxis of physiological and/or pathophysiological conditions in mammals, preferably humans, that are mediated by GHS receptors. The present invention further provides GHS receptor antagonists and agonists that can be used for modulation of these receptors and are useful for treating above conditions, in particular growth retardation, cachexia, short-, medium- and/or long term regulation of energy balance; short-, medium- and/or long term regulation (stimulation and/or inhibition) of food intake; adipogenesis, adiposity and/or obesity; body weight gain and/or reduction; diabetes, diabetes type I, diabetes type II, tumor cell proliferation; inflammation, inflammatory effects, gastric postoperative ileus, postoperative ileus and/or gastrectomy (ghrelin replacement therapy)'. |
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372-MUMNP-2008-ASSIGNMENT(9-1-2012).pdf
372-mumnp-2008-claims(27-2-2008).pdf
372-MUMNP-2008-CLAIMS(AMENDED)-(3-12-2012).pdf
372-MUMNP-2008-CLAIMS(AMENDED)-(9-1-2012).pdf
372-MUMNP-2008-CLAIMS(MARKED COPY)-(3-12-2012).pdf
372-MUMNP-2008-CLAIMS(MARKED COPY)-(9-1-2012).pdf
372-MUMNP-2008-CORRESPONDENCE(19-6-2009).pdf
372-mumnp-2008-correspondence-others.pdf
372-mumnp-2008-correspondence-received.pdf
372-mumnp-2008-description (complete).pdf
372-mumnp-2008-description(complete)-(27-2-2008).pdf
372-MUMNP-2008-FORM 13(9-1-2012).pdf
372-MUMNP-2008-FORM 18(19-6-2009).pdf
372-mumnp-2008-form 2(27-2-2008).pdf
372-mumnp-2008-form 2(title page)-(27-2-2008).pdf
372-MUMNP-2008-FORM 26(9-1-2012).pdf
372-MUMNP-2008-FORM 3(9-1-2012).pdf
372-mumnp-2008-form-pct-ib-306.pdf
372-mumnp-2008-form-pct-ipea-409.pdf
372-mumnp-2008-form-pct-ro-101.pdf
372-mumnp-2008-form-pct-separate sheet-409.pdf
372-MUMNP-2008-PETITION UNDER RULE 137(9-1-2012).pdf
372-MUMNP-2008-REPLY TO EXAMINATION REPORT(9-1-2012).pdf
372-MUMNP-2008-REPLY TO HEARING(3-12-2012).pdf
372-mumnp-2008-wo international publication report(27-2-2008).pdf
Patent Number | 254746 | |||||||||||||||||||||
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Indian Patent Application Number | 372/MUMNP/2008 | |||||||||||||||||||||
PG Journal Number | 51/2012 | |||||||||||||||||||||
Publication Date | 21-Dec-2012 | |||||||||||||||||||||
Grant Date | 14-Dec-2012 | |||||||||||||||||||||
Date of Filing | 27-Feb-2008 | |||||||||||||||||||||
Name of Patentee | UNIVERSITY OF MONTPELLIER I | |||||||||||||||||||||
Applicant Address | 5, BOULEVARD HENRI IV BP 107, F-34006 MONTPELLIER CEDEX 5 | |||||||||||||||||||||
Inventors:
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PCT International Classification Number | A61K31/4196,A61P5/08 | |||||||||||||||||||||
PCT International Application Number | PCT/EP2006/007945 | |||||||||||||||||||||
PCT International Filing date | 2006-08-11 | |||||||||||||||||||||
PCT Conventions:
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