Title of Invention

NOVEL TRIAZOLE DERIVATIVES RECEPTORS

Abstract The present invention provides novel triazole derivatives as ghrelin analogue ligands of growth hormone secretagogue receptors according to formula (I) that are useful in the treatment or prophylaxis of physiological and/or pathophysiological conditions in mammals, preferably humans, that are mediated by GHS receptors. The present invention further provides GHS receptor antagonists and agonists that can be used for modulation of these receptors and are useful for treating above conditions, in particular growth retardation, cachexia, short-, medium- and/or long term regulation of energy balance; short-, medium- and/or long term regulation (stimulation and/or inhibition) of food intake; adipogenesis, adiposity and/or obesity; body weight gain and/or reduction; diabetes, diabetes type I, diabetes type II, tumor cell proliferation; inflammation, inflammatory effects, gastric postoperative ileus, postoperative ileus and/or gastrectomy (ghrelin replacement therapy)'.
Full Text

Documents:

372-mumnp-2008-abstract.pdf

372-MUMNP-2008-ASSIGNMENT(9-1-2012).pdf

372-mumnp-2008-claims(27-2-2008).pdf

372-MUMNP-2008-CLAIMS(AMENDED)-(3-12-2012).pdf

372-MUMNP-2008-CLAIMS(AMENDED)-(9-1-2012).pdf

372-MUMNP-2008-CLAIMS(MARKED COPY)-(3-12-2012).pdf

372-MUMNP-2008-CLAIMS(MARKED COPY)-(9-1-2012).pdf

372-mumnp-2008-claims.pdf

372-MUMNP-2008-CORRESPONDENCE(19-6-2009).pdf

372-mumnp-2008-correspondence-others.pdf

372-mumnp-2008-correspondence-received.pdf

372-mumnp-2008-description (complete).pdf

372-mumnp-2008-description(complete)-(27-2-2008).pdf

372-mumnp-2008-drawings.pdf

372-MUMNP-2008-FORM 13(9-1-2012).pdf

372-MUMNP-2008-FORM 18(19-6-2009).pdf

372-mumnp-2008-form 2(27-2-2008).pdf

372-mumnp-2008-form 2(title page)-(27-2-2008).pdf

372-MUMNP-2008-FORM 26(9-1-2012).pdf

372-MUMNP-2008-FORM 3(9-1-2012).pdf

372-mumnp-2008-form-1.pdf

372-mumnp-2008-form-2.pdf

372-mumnp-2008-form-3.pdf

372-mumnp-2008-form-5.pdf

372-mumnp-2008-form-pct-ib-306.pdf

372-mumnp-2008-form-pct-ipea-409.pdf

372-mumnp-2008-form-pct-ro-101.pdf

372-mumnp-2008-form-pct-separate sheet-409.pdf

372-MUMNP-2008-PETITION UNDER RULE 137(9-1-2012).pdf

372-MUMNP-2008-REPLY TO EXAMINATION REPORT(9-1-2012).pdf

372-MUMNP-2008-REPLY TO HEARING(3-12-2012).pdf

372-mumnp-2008-wo international publication report(27-2-2008).pdf


Patent Number 254746
Indian Patent Application Number 372/MUMNP/2008
PG Journal Number 51/2012
Publication Date 21-Dec-2012
Grant Date 14-Dec-2012
Date of Filing 27-Feb-2008
Name of Patentee UNIVERSITY OF MONTPELLIER I
Applicant Address 5, BOULEVARD HENRI IV BP 107, F-34006 MONTPELLIER CEDEX 5
Inventors:
# Inventor's Name Inventor's Address
1 PERRISSOUD, DANIEL WILHELM-MEISTER-STRASSE 7, 61348 BAD HOMBURG
2 MARTINEZ, JEAN LE JARDIN DES MUSES, 9, RUE JEAN MOULIN, F-34720 CAUX
3 MOULIN ALINE 12, ROUTE DE BEAUVALLON, F-26800 PORTES-LES-VALENCE
4 FEHRENTZ, JEAN-ALAIN 217, AVENUE DE I'ABRIVADO F-3440 ST.NAZAIRE DE PEZAN
5 BOEGLIN, DAMIEN 11, RUE DES PINSONS, F-68420 EGUISHEIM
6 DEMANGE, LUC 14, RUE BUFFON, F-91400 ORSAY
PCT International Classification Number A61K31/4196,A61P5/08
PCT International Application Number PCT/EP2006/007945
PCT International Filing date 2006-08-11
PCT Conventions:
# PCT Application Number Date of Convention Priority Country
1 60/707,941 2005-08-15 U.S.A.
2 05017732.8 2005-08-16 U.S.A.
3 60/787,543 2006-03-31 U.S.A.