Title of Invention

AMINOALCOHOL DERIVATIVES

Abstract The present invention relates to a compound of the formula [I]: wherein (a), in which -Y<SUB>6</SUB></sub> area R<sub>5</sub> each as defined in the description, etc., R<sub>1</sub> is hydrogen, halogen, lower alkyl, hydroxy, etc., R<sub>2</sub> is hydrogen, lower alkyl or hydroxy(lower)alkyl, R<sub>3</sub> is hydrogen or an amino protective group, 20 R<sub>7</sub> is hydrogen, lower alkyl, cyclo(lower)alkyl, lower R9 alkenyl, -Z-R<sub>9</sub> or (b), in which -Z- is -0-, -S-, R<sub>9</sub> -SO- or -SO<sub>2</sub>-, and each R<sub>9</sub> is independently hydrogen, lower alkyl, cyclo(lower)alkyl, etc., and R<sub>8</sub> is -D-E-R<sub>10</sub>, in which -D- is -CONHSO<sub>2</sub>- or -S0<sub>2</suB>NHCO-, E is bond or lower alkylene, and R<sub>10</sub> is halogen, cyano, carboxy, etc., or a prodrug thereof or a salt thereof. The compound [I] of the present invention and pharmaceutically acceptable salts thereof are useful for the prophylactic and/or the therapeutic treatment of ulcer, overactive bladder, and the like.
Full Text

Documents:

1176-CHENP-2007 AMENDED CLAIMS 09-04-2014.pdf

1176-CHENP-2007 AMENDED PAGES OF SPECIFICATION 09-04-2014.pdf

1176-CHENP-2007 CORRESPONDENCE OTHERS 15-10-2013.pdf

1176-CHENP-2007 CORRESPONDENCE OTHERS 12-06-2013.pdf

1176-chenp-2007 correspondence others 20-09-2007.pdf

1176-chenp-2007 correspondence others 21-03-2007.pdf

1176-chenp-2007 form-1 21-03-2007.pdf

1176-CHENP-2007 FORM-3 15-10-2013.pdf

1176-chenp-2007 form-3 21-03-2007.pdf

1176-chenp-2007 form-5 21-03-2007.pdf

1176-CHENP-2007 EXAMINATION REPORT REPLY RECEIVED 09-04-2014.pdf

1176-CHENP-2007 FORM-18.pdf

1176-CHENP-2007 POWER OF ATTORNEY 09-04-2014.pdf

1176-CHENP-2007 PRIORITY DOCUMENT 09-04-2014.pdf

1176-chenp-2007 abstract 21-03-2007.pdf

1176-chenp-2007 claims 21-03-2007.pdf

1176-chenp-2007 description(complete) 21-03-2007.pdf

1176-chenp-2007 description(complete) -1 21-03-2007.pdf

1176-chenp-2007 form-2 21-03-2007.pdf

1176-chenp-2007 form-3 20-09-2007.pdf

1176-chenp-2007 pct 21-03-2007.pdf

1562-2007-AnnexureTo Form 3.pdf

1562-2007-Petition 137 Annex Form 3.pdf


Patent Number 261055
Indian Patent Application Number 1176/CHENP/2007
PG Journal Number 23/2014
Publication Date 06-Jun-2014
Grant Date 31-May-2014
Date of Filing 21-Mar-2007
Name of Patentee ASTELLAS PHARMA INC
Applicant Address 3-11, NIHONBASHI-HONCHO 2-CHOME CHUO-KU TOKYO 103-8411
Inventors:
# Inventor's Name Inventor's Address
1 HATTORI, KOUJI C/O ASTELLAS PHARMA INC 3-11 NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411 JAPAN
2 TODA, SUSUMU C/O ASTELLAS PHARMA INC 3-11 NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411 JAPAN
3 WASHIZUKA, KENICHI C/O ASTELLAS PHARMA INC 3-11 NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411 JAPAN
4 ITO, SHINJI C/O ASTELLAS PHARMA INC 3-11 NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411 JAPAN
5 TANABE, DAISUKE C/O ASTELLAS PHARMA INC 3-11 NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411 JAPAN
6 ARAKI, TAKANOBU C/O ASTELLAS PHARMA INC 3-11 NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411 JAPAN
7 SAKURAI, MINORU C/O ASTELLAS PHARMA INC 3-11 NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411 JAPAN
PCT International Classification Number C07D 213/38
PCT International Application Number PCT/JP05/17669
PCT International Filing date 2005-09-20
PCT Conventions:
# PCT Application Number Date of Convention Priority Country
1 2005900789 2005-02-21 Australia
2 2004905450 2004-09-21 Australia