Title of Invention | AMINOALCOHOL DERIVATIVES |
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Abstract | The present invention relates to a compound of the formula [I]: wherein (a), in which -Y<SUB>6</SUB></sub> area R<sub>5</sub> each as defined in the description, etc., R<sub>1</sub> is hydrogen, halogen, lower alkyl, hydroxy, etc., R<sub>2</sub> is hydrogen, lower alkyl or hydroxy(lower)alkyl, R<sub>3</sub> is hydrogen or an amino protective group, 20 R<sub>7</sub> is hydrogen, lower alkyl, cyclo(lower)alkyl, lower R9 alkenyl, -Z-R<sub>9</sub> or (b), in which -Z- is -0-, -S-, R<sub>9</sub> -SO- or -SO<sub>2</sub>-, and each R<sub>9</sub> is independently hydrogen, lower alkyl, cyclo(lower)alkyl, etc., and R<sub>8</sub> is -D-E-R<sub>10</sub>, in which -D- is -CONHSO<sub>2</sub>- or -S0<sub>2</suB>NHCO-, E is bond or lower alkylene, and R<sub>10</sub> is halogen, cyano, carboxy, etc., or a prodrug thereof or a salt thereof. The compound [I] of the present invention and pharmaceutically acceptable salts thereof are useful for the prophylactic and/or the therapeutic treatment of ulcer, overactive bladder, and the like. |
Full Text |
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1176-CHENP-2007 AMENDED CLAIMS 09-04-2014.pdf
1176-CHENP-2007 AMENDED PAGES OF SPECIFICATION 09-04-2014.pdf
1176-CHENP-2007 CORRESPONDENCE OTHERS 15-10-2013.pdf
1176-CHENP-2007 CORRESPONDENCE OTHERS 12-06-2013.pdf
1176-chenp-2007 correspondence others 20-09-2007.pdf
1176-chenp-2007 correspondence others 21-03-2007.pdf
1176-chenp-2007 form-1 21-03-2007.pdf
1176-CHENP-2007 FORM-3 15-10-2013.pdf
1176-chenp-2007 form-3 21-03-2007.pdf
1176-chenp-2007 form-5 21-03-2007.pdf
1176-CHENP-2007 EXAMINATION REPORT REPLY RECEIVED 09-04-2014.pdf
1176-CHENP-2007 POWER OF ATTORNEY 09-04-2014.pdf
1176-CHENP-2007 PRIORITY DOCUMENT 09-04-2014.pdf
1176-chenp-2007 abstract 21-03-2007.pdf
1176-chenp-2007 claims 21-03-2007.pdf
1176-chenp-2007 description(complete) 21-03-2007.pdf
1176-chenp-2007 description(complete) -1 21-03-2007.pdf
1176-chenp-2007 form-2 21-03-2007.pdf
1176-chenp-2007 form-3 20-09-2007.pdf
1176-chenp-2007 pct 21-03-2007.pdf
1562-2007-AnnexureTo Form 3.pdf
1562-2007-Petition 137 Annex Form 3.pdf
Patent Number | 261055 | ||||||||||||||||||||||||
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Indian Patent Application Number | 1176/CHENP/2007 | ||||||||||||||||||||||||
PG Journal Number | 23/2014 | ||||||||||||||||||||||||
Publication Date | 06-Jun-2014 | ||||||||||||||||||||||||
Grant Date | 31-May-2014 | ||||||||||||||||||||||||
Date of Filing | 21-Mar-2007 | ||||||||||||||||||||||||
Name of Patentee | ASTELLAS PHARMA INC | ||||||||||||||||||||||||
Applicant Address | 3-11, NIHONBASHI-HONCHO 2-CHOME CHUO-KU TOKYO 103-8411 | ||||||||||||||||||||||||
Inventors:
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PCT International Classification Number | C07D 213/38 | ||||||||||||||||||||||||
PCT International Application Number | PCT/JP05/17669 | ||||||||||||||||||||||||
PCT International Filing date | 2005-09-20 | ||||||||||||||||||||||||
PCT Conventions:
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