| Title of Invention | AZEPINOINDOLE DERIVATIVES AS PHARMACEUTICAL AGENTS |
|---|---|
| Abstract | Compounds for use in pharmaceutical compositions and methods for modulating the activity of nuclear receptors are provided. In particular, compounds for use in compositions and methods for modulating the farnesoid X receptor, and/or orphan nuclear receptors, are provided.: formula (I) or a pharmaceutically acceptable derivative thereof; wherein: R1 is -C(J)OR14, -C(J)SR14 and -C(J)N(R15)R16, J is O, S or NR17, R2 is hydrogen, halo or optionally substituted alkyl; R3 is -C(O)R9, R4, R5, R6 and R7 and R8 are as described in the claims. |
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01497-kolnp-2006-assignment.pdf
01497-kolnp-2006-correspondence other.pdf
01497-kolnp-2006-correspondence others-1.1.pdf
01497-kolnp-2006-correspondence.pdf
01497-kolnp-2006-description complete.pdf
01497-kolnp-2006-form-3-1.1.pdf
01497-kolnp-2006-international publication.pdf
01497-kolnp-2006-international search report.pdf
01497-kolnp-2006-priority document.pdf
1497-KOLNP-2006-(04-07-2013)-CORRESPONDENCE.pdf
1497-KOLNP-2006-(10-09-2014)-ABSTRACT.pdf
1497-KOLNP-2006-(10-09-2014)-CLAIMS.pdf
1497-KOLNP-2006-(10-09-2014)-CORRESPONDENCE.pdf
1497-KOLNP-2006-(10-09-2014)-FORM-2.pdf
1497-KOLNP-2006-(10-09-2014)-MARKEDUP COPY.pdf
1497-KOLNP-2006-AMANDED CLAIMS.pdf
1497-KOLNP-2006-ASSIGNMENT.pdf
1497-KOLNP-2006-CORRESPONDENCE 1.1.pdf
1497-KOLNP-2006-CORRESPONDENCE 1.2.pdf
1497-KOLNP-2006-DESCRIPTION (COMPLETE).pdf
1497-KOLNP-2006-EXAMINATION REPORT REPLY RECIEVED.pdf
1497-KOLNP-2006-EXAMINATION REPORT.pdf
1497-KOLNP-2006-FORM 3 1.1.pdf
1497-KOLNP-2006-GRANTED-ABSTRACT.pdf
1497-KOLNP-2006-GRANTED-CLAIMS.pdf
1497-KOLNP-2006-GRANTED-DESCRIPTION (COMPLETE).pdf
1497-KOLNP-2006-GRANTED-DRAWINGS.pdf
1497-KOLNP-2006-GRANTED-FORM 1.pdf
1497-KOLNP-2006-GRANTED-SPECIFICATION.pdf
1497-KOLNP-2006-INTERNATIONAL PUBLICATION.pdf
1497-KOLNP-2006-INTERNATIONAL SEARCH REPORT.pdf
1497-KOLNP-2006-OTHERS 1.1.pdf
1497-KOLNP-2006-OTHERS PCT FORM.pdf
1497-KOLNP-2006-PCT REQUEST FORM.pdf
1497-KOLNP-2006-PETITION UNDER RULE 137.pdf
1497-KOLNP-2006-REPLY TO EXAMINATION REPORT.pdf
1497-KOLNP-2006-TRANSLATED COPY OF PRIORITY DOCUMENT.pdf
| Patent Number | 262950 | ||||||||||||||||||||||||
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| Indian Patent Application Number | 1497/KOLNP/2006 | ||||||||||||||||||||||||
| PG Journal Number | 40/2014 | ||||||||||||||||||||||||
| Publication Date | 03-Oct-2014 | ||||||||||||||||||||||||
| Grant Date | 25-Sep-2014 | ||||||||||||||||||||||||
| Date of Filing | 01-Jun-2006 | ||||||||||||||||||||||||
| Name of Patentee | EXELIXIS, INC. | ||||||||||||||||||||||||
| Applicant Address | 170 HARBOUR WAY, P.O.BOX 511, SOUTH SAN FRANCISCO, CALIFORNIA 94083-0511 | ||||||||||||||||||||||||
Inventors:
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| PCT International Classification Number | C07D 487/04 | ||||||||||||||||||||||||
| PCT International Application Number | PCT/US2004/040352 | ||||||||||||||||||||||||
| PCT International Filing date | 2004-12-01 | ||||||||||||||||||||||||
PCT Conventions:
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