| Title of Invention | 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5-(HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS |
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| Abstract | The present invention provides a compound having a superior acid secretion inhibitory effect and showing antiulcer activity and the like. The present invention provides a compound represented by the formula (I) wherein R1 is a nitrogen- containing monocyclic heterocyclic group optionally condensed with a benzene ring or a heterocyclic optionally has substituent(s), R2 is an optionally substituted C6-14 aryl group, an optionally substituted thienyl group or an optionally substituted pyridyl group, R3 and R4 are each a hydrogen atom, or one of R3 and R4 is a hydrogen atom and the optionally substituted tower alkyl group, an acyl group, a halogen atom, a cyano group or a nitro group, and R3 is an alkyl group or a salt thereof. |
| Full Text | The present invention provides a compound having a superior acid secretion inhibitory effect and showing antiulcer activity and the like. The present invention provides a compound represented by the formula (I) wherein R1 is a nitrogen- containing monocyclic heterocyclic group optionally condensed with a benzene ring or a heterocyclic optionally has substituent(s), R2 is an optionally substituted C6-14 aryl group, an optionally substituted thienyl group or an optionally substituted pyridyl group, R3 and R4 are each a hydrogen atom, or one of R3 and R4 is a hydrogen atom and the optionally substituted tower alkyl group, an acyl group, a halogen atom, a cyano group or a nitro group, and R3 is an alkyl group or a salt thereof. |
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01285-kolnp-2008-correspondence others.pdf
01285-kolnp-2008-international search report.pdf
01285-kolnp-2008-pct priority document notification.pdf
01285-kolnp-2008-pct request form.pdf
1285-KOLNP-2008-(01-02-2013)-ANNEXURE TO FORM 3.pdf
1285-KOLNP-2008-(01-02-2013)-CORRESPONDENCE.pdf
1285-KOLNP-2008-(01-02-2013)-OTHERS-1.pdf
1285-KOLNP-2008-(01-02-2013)-OTHERS.pdf
1285-KOLNP-2008-(07-05-2013)-ABSTRACT.pdf
1285-KOLNP-2008-(07-05-2013)-ANNEXURE TO FORM 3.pdf
1285-KOLNP-2008-(07-05-2013)-CLAIMS.pdf
1285-KOLNP-2008-(07-05-2013)-CORRESPONDENCE.pdf
1285-KOLNP-2008-(07-05-2013)-OTHERS.pdf
1285-KOLNP-2008-(07-05-2013)-PETITION UNDER RULE 137.pdf
1285-KOLNP-2008-(22-07-2013)-ANNEXURE TO FORM 3.pdf
1285-KOLNP-2008-(22-07-2013)-CORRESPONDENCE.pdf
1285-KOLNP-2008-(25-08-2009)-FORM 13.pdf
1285-KOLNP-2008-CORRESPONDENCE-1.1.pdf
| Patent Number | 264318 | ||||||||||||
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| Indian Patent Application Number | 1285/KOLNP/2008 | ||||||||||||
| PG Journal Number | 52/2014 | ||||||||||||
| Publication Date | 26-Dec-2014 | ||||||||||||
| Grant Date | 22-Dec-2014 | ||||||||||||
| Date of Filing | 31-Mar-2008 | ||||||||||||
| Name of Patentee | TAKEDA PHARMACEUTICAL COMPANY LIMITED | ||||||||||||
| Applicant Address | 1-1, DOSHOMACHI 4-CHOME, CHUO-KU, OSAKA-SHI, OSAKA | ||||||||||||
Inventors:
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| PCT International Classification Number | C07D 207/48 | ||||||||||||
| PCT International Application Number | PCT/JP2006/317408 | ||||||||||||
| PCT International Filing date | 2006-08-29 | ||||||||||||
PCT Conventions:
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